托帕利酯
| CAS号 | 74163-84-1 | 货号 | BCP18912 |
| 中文名 | 托帕利酯 | ||
| 英文名 | Troparil | ||
| 中文别名 | |||
| 英文别名 | (–)-2β-Carbomethoxy-3β-phenyltropane; WIN 35,065-2; β-CPT; | ||
| 分子式 | C16H21NO2 | 分子量 | 259.34 |
| 生物活性 | Troparil (also known as (–)-2β-Carbomethoxy-3β-phenyltropane, WIN 35,065-2, or β-CPT) is a stimulant drug used in scientific research. Troparil is a phenyltropane-based dopamine reuptake inhibitor (DRI) that is derived from methylecgonidine. Troparil is a few times more potent than cocaine as a dopamine reuptake inhibitor, but is less potent as a serotonin reuptake inhibitor,and has a duration spanning a few times longer, since the phenyl ring is directly connected to the tropane ring through a non-hydrolyzable carbon-carbon bond. The lack of an ester linkage removes the local anesthetic action from the drug, so troparil is a pure stimulant. This change in activity also makes troparil slightly less cardiotoxic than cocaine. The most commonly used form of troparil is the tartrate salt, but the hydrochloride and naphthalenedisulfonate salts are also available, as well as the free base. | ||
| 信号通路 | Neuro Signaling Pathway GPCR/G Protein | ||
| 靶 点 | Dopamine Receptor | ||
结构式
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